Carvedilol is a pharmaceutical agent classified as a non-selective beta-blocker and alpha-1 blocker. Healthcare providers use it in the treatment of various cardiovascular conditions, primarily heart failure and hypertension.Carvedilol exerts its therapeutic effects by blocking both beta receptors in the heart (particularly beta-1 receptors) and alpha-1 receptors in blood vessels. …
Atenolol: Mechanism of Action, Uses, Side Effects, Stability, and Storage
Atenolol is a medication that belongs to the class of drugs known as beta-blockers. It is commonly prescribed for the treatment of cardiovascular conditions, particularly hypertension (high blood pressure) and angina (chest pain). Atenolol works by selectively blocking beta-1 adrenergic receptors in the heart. Doing so reduces the effects of …
Propranolol: Mechanism, Uses, Side effects
Propranolol is a medication belonging to the class of drugs known as beta-adrenergic blockers. It is a non-selective beta blocker, which blocks beta-1 (β1) and beta-2 (β2) adrenergic receptors. Propranolol affects receptors primarily found in the heart, blood vessels, and lungs. Healthcare providers use it for various cardiovascular and non-cardiovascular …
Beta-adrenergic blockers
Beta-adrenergic blockers, often simply referred to as beta blockers, are a class of medications that block the effects of adrenaline (epinephrine) and related hormones. These drugs primarily target beta-adrenergic receptors, which are found in various tissues, including the heart, blood vessels, and certain parts of the nervous system. Beta-blockers exert …
Prazosin: Mechanism, Uses, Side effects
Prazosin is a medication classified as an alpha-1 adrenergic blocker. It belongs to the class of drugs known as alpha-adrenergic antagonists. Prazosin primarily acts on alpha-1 receptors, blocking the effects of norepinephrine and leading to vasodilation and relaxation of smooth muscle in blood vessels. Here are key points about prazosin: …
Phenoxybenzamine: Mechanism, Uses, Side effects
Phenoxybenzamine is a medication classified as an alpha-adrenergic antagonist, specifically an irreversible alpha-blocker. It is used primarily to treat conditions associated with excessive sympathetic nervous system activity, such as pheochromocytoma, a rare adrenal tumor that releases high levels of catecholamines, leading to severe hypertension. Here are key points about phenoxybenzamine: …
Phentolamine: Mechanism, Uses, Side effects
Phentolamine is a medication classified as an alpha-adrenergic antagonist, specifically an alpha-blocker. It acts by blocking the effects of norepinephrine and other similar neurotransmitters at alpha-adrenergic receptors. Phentolamine is a non-selective alpha-blocker, meaning it blocks both alpha-1 and alpha-2 receptors. Here are key points about phentolamine: 1. Mechanism of Action …
Tolazoline: Mechanism, Uses, Side effects
Tolazoline is a medication that belongs to the class of drugs known as alpha-adrenergic blockers. It is primarily used as a vasodilator, which relaxes and widens blood vessels. This vasodilatory effect is attributed to its ability to block alpha-adrenergic receptors. Here are some key points about tolazoline: Mechanism of Action …
Adrenergic antagonists/adrenergic blockers/adrenergic receptor antagonists
Adrenergic antagonists, also known as adrenergic blockers or adrenergic receptor antagonists, are a class of drugs that interfere with the actions of the sympathetic nervous system, specifically by blocking the effects of neurotransmitters like norepinephrine and epinephrine (adrenaline) at adrenergic receptors. These receptors are found throughout the body and are …